Tamoxifen in bodybuilding is widely used in conjunction with anbolic steroids for the prevention and treatment of gynecomastia – the growth of the female breast. Below we will talk about how the drug against breast cancer got into the pharmacological first-aid kits of modern bodybuilders, about the mechanism of action and effectiveness of tamoxifen on the PCT cycle, what are the side effects as well as where to buy tamoxifen online?
What is Tamoxifen?
Tamoxifen citrate is a pharmacological drug that acts on the receptors of estrogen (female sex hormone) in organism, suppressing its action.
It was created in 1961. The most common form of tamoxifen is tamoxifen citrate, and the most famous brand is Nolvadex.
Often referred to as an antiestrogen, tamoxifen citrate is actually both an antagonist and an agonist. This means that it acts as an antiestrogen in some areas of the body and as estrogen in others.
In medicine, tamoxifen has been used for several decades for the treatment of breast cancer and is recognized as one of the most effective drugs.
In bodybuilding, tamoxifen is used by anabolic steroid users during and after anabolic steroids (PCT) to combat gynecomastia (female breast growth), one of the many side effects of steroids.
How does tamoxifen work?
Tamoxifen acts as an antagonist and agonist towards the hormone estrogen.
Its anti-estrogenic properties are manifested in the fact that it acts on the estrogen receptors in certain parts of the body, making them insensitive to estrogen. This applies primarily to the cells of the mammary glands (breast).
This explains its effectiveness in the fight against breast cancer, as this type of cancer feeds on “estrogen”.
In bodybuilding, tamoxifen inhibits breast growth, which is also due to an increase in estrogen levels due to the partial conversion of testosterone / steroids to estrogen.
With the antiestrogenic effect of tamoxifen, everything is more or less clear. It is more difficult to understand its action as estrogen in other parts of the body.
Tamoxifen citrate works like estrogen in the liver. Is it good or bad?
On one of the sites selling sports pharmacology, the opinion is voiced that the estrogenic activity of tamoxifen associated with the liver improves the state of the cardiovascular system, in particular, reduces the level of cholesterol in the blood …
If so, then this is an undoubted advantage for those bodybuilders who use steroids, since they have a negative effect on cholesterol, blood vessels “clogged”.
Tamoxifen in bodybuilding on steroid cycle
In bodybuilding, tamoxifen is taken both on and after the steroid cycle (PCT). More often – after.
Some types of steroids – nandrolone and testosterone – increase estrogen levels, as they are partially converted into it during metabolism by the aromatase enzyme.
When estrogen grows, the likelihood of breast growth naturally increases, and more water is retained in the body, which can lead to an increase in blood pressure.
What tamoxifen does and why bodybuilders take it: It does NOT lower estrogen levels, but blocks the receptors of this hormone in the breast (makes them immune). Accordingly, it has no effect on water retention and other possible side effects of elevated female sex hormone levels …
Does tamoxifen guarantee complete protection against gynecomastia? No. It depends on estrogen levels and genetic characteristics.
If tamoxifen does not help, then stronger protection is needed in the form of aromatase inhibitors, which prevent the conversion of testosterone into estrogen … Or maybe it’s just time to think about what the hell are you doing …
What are the positive effects of tamoxifen? How tamoxifen affects the body
Tamoxifen is characterized by neither androgenic nor anabiotic effects on the body. Many steroids have a tendency to convert estrogens into female sex hormones, and it is this process that tamoxifen prevents.
It is worth noting that this antiestrogen blocks the functioning of all estrogen receptors in the athlete’s body. Unlike another, also quite popular anti-estrogen, clomid, which interferes with the work of estrogen receptors only in the pituitary gland and testes.
Next, we will consider in more detail the questions about the effect of tamoxifen on different groups of organs and body systems:
How tamoxifen affects potency – the anti-estrogen can even be used as a testosterone booster in post-cycle therapy. It significantly increases the concentration of natural male sex hormone in the body – for ten days of daily intake of tamoxifen 20 mg, it can increase testosterone levels by 42%. As a result, an athlete can observe an increase in potency, increased libido, sexual activity, which has a beneficial effect on the quality of sexual life.
How tamoxifen affects the blood – almost immediately after taking the pill, you can observe that the concentration of cholesterol in the blood significantly increases, which has a positive effect on the Work of the heart. Also, the effect of antiestrogen can significantly reduce the risk of developing atherosclerosis, and has prophylaxis against cardiovascular diseases.
How tamoxifen affects the liver – tamoxifen significantly improves liver function. Damage to this organ is observed only in the case of existing diseases that have been exacerbated by the intake of an antiestrogen – hepatitis and other serious liver diseases.
The antiestrogenic effect of the drug on the athlete’s body is based on blocking the functioning of estrogen receptors, and not, as many think, a complete cessation of the conversion of testosterone into estrogens.
Antiestrogen does not completely prevent estrogenic activity, but only inhibits it.
Also, in addition to the above effects, the drug has the following positive effects on the athlete’s body:
- an increase in strength capabilities;
- an increase in muscle volume, which makes the drug quite popular in bodybuilding, and in sports there is an opinion that no victory at the championships can do without this antiestrogen;
- pronounced drawing of the relief of the muscles, increasing the hardness of the muscles;
- strong antiestrogenic effect, which made tamoxifen quite popular in bodybuilding, it is one of the main drugs during post-cycle therapy;
- disposal of excess subcutaneous fat deposits;
- prevention of feminization.
It is worth noting that tamoxifen cannot be used with every anabolic and androgenic agent. It is contraindicated to take it on a course or after a course of nandrolones and trenbolones.
These steroids have progestogenic activity and tamoxifen tends to increase it significantly, which can lead to serious adverse reactions.
In this case, tamoxifen is successfully replaced with clomid.The highest concentration of estrogens in the body during the course of anabolic and androgenic steroids is observed at the end of the first week of administration, therefore, tamoxifen is used on the course starting from the second week. In post-cycle therapy, they begin to take it after the active component of the anabolic agent ceases to act in the body. It is recommended to buy tamoxifen online for best offers also you can analyse the product quality with the reviews posted by the customers.